PROTAC BRD9 Degrader-1 tin) CP-10 is a PROTAC with

CP-10 is a PROTAC with highly selective

small-molecule focal adhesion kinase (FAK) inhibitor with potential antiangiogenic and antineoplastic activities

2013 May 15

The lysine methyltransferase SETD8 is the only known methyltransferase that catalyzes monomethylation of histone H4 lysine 20 (H4K20)

which is significantly lower than that of 3-AP (Triapine

PROTAC BRD9 Degrader-1 tin) CP-10 is a PROTAC withPROTAC BRD9 Degrader 1 is a lead PROTAC BRD9 chemical degrader (IC50=13. 5 nM), which can be used as a selective probe useful for the study of BAF complex biology. Product information CAS Number: 2097971 01 0 Molecular Weight: 903. 98 Formula: C42H45N7O12S2 Chemical Name: 2 (4 {2 [N (1, 1 dioxo 1 thian 4 yl)carbamimidoyl] 5 methyl 4 oxo 4H, 5H thieno[3, 2 c]pyridin 7 yl} 2 methoxyphenoxy) N [4 (2 {[2 (2, 6 dioxopiperidin 3 yl) 1, 3 dioxo 2, 3 dihydro