Setiptiline Size:Solid 10 mg InChi: InChI=1S/C12H15N3O2/c1-14-5-7-15(8-6-14)10-4-2-3-9-11(10)17-12(16)13-9/h2-4H

InChi: InChI=1S/C12H15N3O2/c1-14-5-7-15(8-6-14)10-4-2-3-9-11(10)17-12(16)13-9/h2-4H

InChi: InChI=1S/C26H19N3O5/c1-25-26(33

is a highly potent and selective inhibitor of Lysine Specific Demethylase 1 (LSD1) with IC50 <20 nM

10058-F4 induces cell-cycle arrest

Solubility: DMSO: 91 mg/mL(201

Setiptiline Size:Solid 10 mg InChi: InChI=1S/C12H15N3O2/c1-14-5-7-15(8-6-14)10-4-2-3-9-11(10)17-12(16)13-9/h2-4HSetiptiline, also known as MO 8282 and teciptiline, is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). It was launched in 1989 for the treatment of depression in Japan by Mochida. Setiptiline acts as a norepinephrine reuptake inhibitor,[3] 2 adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5 HT2A, 5 HT2C, and or 5 HT3 subtypes, as well as an H1 receptor